Does adrafinil feel the same as modafinil?
Adrafinil is a prodrug; it is primarily metabolized in vivo to modafinil, resulting in very similar pharmacological effects. Unlike modafinil, however, it takes time for the metabolite to accumulate to active levels in the bloodstream….Adrafinil.
Clinical data | |
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Identifiers | |
show IUPAC name | |
CAS Number | 63547-13-7 |
PubChem CID | 3033226 |
How long does it take for adrafinil to convert to modafinil?
Its half-life is 11 to 14 hours. Up to 60% of modafinil is converted into modafinil acid and modafinil sulfone, both of which are inactive metabolites. Metabolism primarily occurs through CYP3A4/5, but the compound has also been reported to induce CYP2C19 in vitro.
What is the closest thing to modafinil?
Armodafinil, sold under the brand name Nuvigil, is a newer drug compared to modafinil. It was approved in 2007 as the R-enantiomer of modafinil.
What are the benefits of adrafinil?
They increase the release of dopamine, serotonin, and norepinephrine. Fatigue is reduced and there is an increase in alertness and improvement in vigilance performance.
How to best use adrafinil?
How to Use Adrafinil. Experts recommend taking Adrafinil at a dose of around 100mg to 300mg daily . While some doses range from 600mg to 1,200mg, it is not advisable to exceed a 600mg dose. Generally, it is best to take Adrafinil upon waking in the morning and on an empty stomach .
Is modafinil and/or armodafinil safe to use?
Both Modafinil and Armodafinil are incredibly effective at mitigating excessive sleepiness. This can be especially beneficial for people suffering from shift work disorder, sleep apnea or narcolepsy. Modafinil, though safe at is may be, does come with its some minor side effects.
Is modafinil bad for the liver?
A very bad and sometimes deadly reaction has happened with modafinil. Most of the time, this reaction has signs like fever, rash, or swollen glands with problems in body organs like the liver, kidney, blood, heart, muscles and joints, or lungs.
Is adrafinil available at GNC?
While Adrafinil is not available for sale at established pharmacies and stores like GNC / Walmart / Walgreens / CVS / Boots UK etc – Adrafinil is available to buy online at official website of Absorb Your Health , who is the market leader of nootropic supplements.